Compile Data Set for Download or QSAR
maximum 50k data
Found 6 of kd data for polymerid = 9742
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50552139(CHEMBL4790706)
Affinity DataKd:  21nMAssay Description:Antagonist activity at AT1 receptor in rat aortic ringsMore data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50587871(CHEMBL5176610)
Affinity DataKd:  21nMAssay Description:Antagonist activity at AT1 receptor in rat aortic ringsMore data for this Ligand-Target Pair
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50543138(CHEMBL4646526)
Affinity DataKd:  65nMAssay Description:Binding affinity to human TLR8 extracellular domain (27 to 827 residues) expressed in Drosophila S2 cells by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50514141(CHEMBL4543348)
Affinity DataKd:  86nMAssay Description:Binding affinity to human TLR8 (27 to 827 residues) expressed in HEK293 cells in presence of R848 by ITC analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50408508(CHEMBL5277457)
Affinity DataKd:  220nMAssay Description:Antagonist activity at AT1 receptor in rat aortic ringsMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetToll-like receptor 8(Homo sapiens (Human))TBA
LigandPNGBDBM50514792(CHEMBL4519240)
Affinity DataKd:  225nMAssay Description:Binding affinity to human TLR8 ectodomain by isothermal titration calorimetryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB